Constrained α/γ-peptides: a new stable extended structure in solution without any hydrogen bond and characterized by a four-fold symmetry.

نویسندگان

  • Francelin Bouillère
  • Debby Feytens
  • Didier Gori
  • Régis Guillot
  • Cyrille Kouklovsky
  • Emeric Miclet
  • Valérie Alezra
چکیده

Small α/γ-peptides alternating α-aminoisobutyric acid and cyclic γ-amino acid residues are described. NMR studies together with restrained simulated annealing revealed that an extended backbone conformation largely dominates in solution for as short as 4-residues long oligomers. This new fold type is devoid of any hydrogen bond and characterized by a four-fold symmetry.

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عنوان ژورنال:
  • Chemical communications

دوره 48 14  شماره 

صفحات  -

تاریخ انتشار 2012